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2019
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Invention
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Compositions comprising enzyme-cleavable amphetamine prodrugs and inhibitors thereof. Pharmaceuti... |
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2016
|
Invention
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Compositions comprising enzyme-cleavable ketone-modified opioid prodrugs and optional inhibitors ... |
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2015
|
Invention
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Active agent prodrugs with heterocyclic linkers.
The embodiments provide prodrug compounds of Fo... |
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|
Invention
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Compositions comprising enzyme-cleavable opioid prodrugs and inhibitors thereof. Pharmaceutical c... |
|
|
Invention
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Compositions comprising enzyme-cleavable oxycodone prodrug. The embodiments provide Compound KC-8... |
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2014
|
Invention
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Controlled release of phenolic opioids.
A method of providing a patient with controlled release ... |
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|
Invention
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Pharmaceutical compositions with attenuated release of phenolic opioids. Pharmaceutical compositi... |
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|
Invention
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Opioid prodrugs with heterocyclic linkers. The embodiments provide prodrug compounds of Formulae ... |
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2012
|
Invention
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Compositions comprising enzyme-cleavable prodrugs of active agents and inhibitors thereof.
The p... |
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|
Invention
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Compositions comprising enzyme-cleavable phenol-modified opioid prodrugs and inhibitors thereof. ... |
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|
Invention
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Controlled release of phenolic opioids. A method of providing a patient with controlled release o... |
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|
Invention
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Active agent prodrugs with heterocyclic linkers. The embodiments provide prodrug compounds of For... |
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|
Invention
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Compositions for reducing risk of adverse events caused by drug-drug interactions.
The present d... |
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|
Invention
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Compositions for reducing risk of adverse events caused by drug-drug interactions. The present di... |
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|
Invention
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Compositions comprising enzyme-cleavable oxycodone prodrug. The embodiments provide Compound KC-7... |
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2011
|
Invention
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Peripheral opioid agonists and peripheral opioid antagonists.
The present disclosure provides co... |
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|
Invention
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Compositions comprising enzyme-cleavable amphetamine prodrugs and inhibitors thereof.
Pharmaceut... |
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|
Invention
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Peripheral opioid agonists and peripheral opioid antagonists. The present disclosure provides com... |
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2010
|
Invention
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Compositions comprising enzyme-cleavable hydromorphone prodrug.
The embodiments provide Compound... |
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Invention
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Compositions comprising enzyme-cleavable phenol-modified tapentadol prodrug. A method of providin... |
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|
Invention
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Compositions comprising enzyme-cleavable hydromorphone prodrug. The embodiments provide Compound ... |
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|
Invention
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Compositions comprising enzyme-cleavable opioid prodrugs and inhibitors thereof.
Pharmaceutical ... |
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|
Invention
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Compositions comprising enzyme-cleavable opioid prodrugs and inhibitors thereof. The present disc... |
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|
Invention
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Compositions comprising enzyme-cleavable prodrugs of active agents and inhibitors thereof. The pr... |
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2009
|
Invention
|
Analogs of propofol, preparation thereof and use as anesthetics.
Compounds of formula (I) wherei... |
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|
Invention
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Anesthetic compounds.
The invention provides novel phenolic ester local anesthetic compounds. Th... |
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2008
|
Invention
|
Peripheral phenolic opioid antagonist.
N-Methyldiprenorphine, useful as an opioid antagonist. |
|
|
Invention
|
Pro-drugs for controlled release of biologically active compounds. Pro-drugs containing an electr... |
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|
Invention
|
N-17-alkylated prodrugs of opioids.
Compounds of formula (II) R1R2R3N+—(C(R1a)(R2a))—Ar—Z—C(O)—Y... |
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|
Invention
|
Prodrugs of peripheral phenolic opioid antagonists.
Compounds of formula (I)
in which X, ... |
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2007
|
Invention
|
Anesthetic compounds.
In one embodiment the invention provides novel compounds of Formula (I) as... |
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2006
|
Invention
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Prodrugs of active agents. Disclosed herein are prodrugs of active agents which contain at least ... |
