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				    							2022
				    							
				    						
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				    							Invention
				    						
				    						
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				    					Immunoglobulin expression levels as biomarker for proteasome inhibitor response. 
Methods of trea... | 
				    				
				    			
				    				
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				    							2021
				    							
				    						
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				    							Invention
				    						
				    						
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				    					Compounds for proteasome enzyme inhibition. 
Peptide-based compounds including heteroatom-contain... | 
				    				
				    			
				    				
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				    							2020
				    							
				    						
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				    							Invention
				    						
				    						
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				    					Tripeptide epoxy ketone protease inhibitors. Provided herein are tripeptide epoxy ketone protease... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Combination therapy with peptide epoxyketones. 
The invention provides combination therapy, where... | 
				    				
				    			
				    				
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				    							2019
				    							
				    						
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				    							Invention
				    						
				    						
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				    					Compounds for proteasome. 
Peptide-based compounds including heteroatom-containing, three-membere... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Peptide epoxyketone proteasome inhibitors in combination with pim kinase inhibitors for treatment... | 
				    				
				    			
				    				
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				    							2018
				    							
				    						
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				    							Invention
				    						
				    						
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				    					Prodrugs of peptide epoxy ketone protease inhibitors. This disclosure features compounds that are... | 
				    				
				    			
				    				
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				    							2017
				    							
				    						
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				    							Invention
				    						
				    						
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				    					Combination therapy with peptide epoxyketones. ABSTRACT The invention provides combination therap... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Peptide epoxyketone immunoproteasome inhibitors. Provided herein are tripeptide epoxy ketone prot... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Compounds for enzyme inhibition. Peptide-based compounds including heteroatom-containing, three-m... | 
				    				
				    			
				    				
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				    							2016
				    							
				    						
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				    							Invention
				    						
				    						
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				    					Combination therapy with peptide epoxyketones. The invention provides combination therapy, wherei... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Modified release formulations for oprozomib. 
This disclosure features modified release pharmaceu... | 
				    				
				    			
				    				
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				    							2015
				    							
				    						
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				    							Invention
				    						
				    						
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				    					Compunds for enzyme inhibition. 
Peptide-based compounds including heteroatom-containing, three-m... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Crystalline tripeptide epoxy ketone protease inhibitors. The invention relates to crystalline tri... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Compounds for enzyme inhibition. One aspect of the invention relates to inhibitors that preferent... | 
				    				
				    			
				    				
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				    							2014
				    							
				    						
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				    							Invention
				    						
				    						
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				    					Use of peptide epoxyketones for metastasis suppression. 
The invention provides a method of repre... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Immunoglobulin expression levels as biomarker for proteasome inhibitor response. Methods of treat... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Dipeptide and tripeptide epoxy ketone protease inhibitors. Provided herein are dipeptide and trip... | 
				    				
				    			
				    				
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				    							2013
				    							
				    						
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				    							Invention
				    						
				    						
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				    					Compounds for enzyme inhibition. 
One aspect of the invention relates to inhibitors that preferen... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Modified release formulations for oprozomib. This disclosure features modified release pharmaceut... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Liposomal compositions of epoxyketone-based proteasome inhibitors. 
Liposomal compositions compri... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Liposomal compositions of epoxyketone-based proteasome inhibitors. Liposomal compositions compris... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Prodrugs of peptide epoxy ketone protease inhibitors. 
This disclosure features compounds that ar... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Prodrugs of peptide epoxy ketone protease inhibitors. Provided herein are compounds of formula (I... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Cyclodextrin complexation methods for formulating peptide proteasome inhibitors. This disclosure ... |