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				    							2025
				    							
				    						
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				    							Invention
				    						
				    						
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				    					Heterocyclic inhibitors of ubiquitin specific protease 1 (usp1) in combination with additional ag... | 
				    				
				    			
				    				
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				    							G/S
				    						
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				    					Computers; Computer software applications, downloadable, for using artificial intelligence for au... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Werner syndrome recq helicase (wrn) inhibitors and methods of uses thereof. Provided compounds, c... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Novel compounds as cyclic gmp-amp synthase inhibitor and uses thereof. Described herein are cycli... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Scalable framework for 3d molecular design via language modeling and reinforcement learning. A co... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Crystalline tead inhibitor and uses thereof. Described herein are crystalline forms of a small mo... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Tead inhibitors and methods of uses thereof. The disclosure provides for compounds and methods fo... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Tead inhibitor combinations and uses thereof. Described herein are methods of treating cancer usi... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Crystalline cyclin-dependent kinase (cdk) 12 and/or cdk13 inhibitor and uses thereof. Described h... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Cyclin-dependent kinase (cdk) 12 and/or cdk13 inhibitor combinations and uses thereof. Described ... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Novel compounds as glucocorticoid receptor modulators and uses thereof. Described herein are gluc... | 
				    				
				    			
				    				
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				    							2024
				    							
				    						
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				    							Invention
				    						
				    						
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				    					Novel compounds as glp-1r agonists and uses thereof. Described herein are GLP-1R agonists and pha... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Methods and systems for alchemical binding free energy. A computer-implemented method can include... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Novel compounds as modulators of sodium channels and uses thereof. Described herein are sodium ch... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Cbl-b inhibitors and methods of uses thereof. Described herein are Casitas B-lineage lymphoma (Cb... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					3cl-protease inhibitors for treating or preventing veterinary coronavirus infections. Provided he... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Novel compounds as pkmyt1 inhibitors and use thereof. Disclosed are compounds or pharmaceutically... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Combinations treatments of diacylglycerol kinase (dgk) alpha inhibitors and other therapies. Desc... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Bifunctional compounds for targeting pkmyt1 and methods of use. Disclosed herein are bifunctional... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Fused ring compound, and preparation method therefor and use thereof. A fused ring compound, and ... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Method and medicament for treating endometriosis. Provided is a method and a medicament for treat... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Ectonucleotide pyrophosphatase-phosphodiesterase 1 (enpp1) inhibitors and uses thereof. Described... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Crytsalline forms of ectonucleotide pyrophosphatase-phosphodiesterase 1 (enpp1) inhibitors and us... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Crystalline beta-lactam derivatives and uses thereof. Described herein are crystalline forms of a... | 
				    				
				    			
				    				
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				    							G/S
				    						
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				    					Downloadable and recorded computer software platforms using artificial intelligence for automated... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Pharmaceutical formulations for inhalation and uses thereof. Provided herein are pharmaceutical f... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Ectonucleotide pyrophosphatase/phosphodiesterase 1 (enpp1) inhibitor combinations and uses thereo... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Crystalline tnik inhibitor and uses thereof. Described herein are crystalline forms of a TNIK inh... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Substituted thiazole compounds as cdk2/4/6 inhibitors and methods of use thereof. The disclosure ... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Synthesis of macrocyclic compound and medical use of macrocyclic compound. Provided in the presen... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Kras inhibitors and uses thereof. KRAS mutation inhibitors and pharmaceutical compositions compri... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Prmt5 inhibitors and uses thereof. Provides for compounds and compositions for modulating or inhi... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Nlrp3 inflammasome inhibitors and uses thereof. Described herein are NOD-like receptor protein 3 ... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Spiro derivatives as wrn inhibitors. Provided compounds of Formula (I) or pharmaceutically accept... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Small molecule inhibitors of ubiquitin specific protease 1 (usp1) and uses thereof. The disclosur... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Prolyl hydroxylase domain-containing protein (phd) inhibitors, combinations and uses thereof. Des... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Crystalline prolyl hydroxylase domain-containing protein (phd) inhibitor and uses thereof. Crysta... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Crystalline prolyl hydroxylase domain-containing protein (phd) inhibitor and uses thereof. Descri... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Crystalline sars-cov-2 inhibitor and uses thereof. Described herein are crystalline forms of a sm... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Crystalline lysine acetyltransferase 6a (kat6a) inhibitor and uses thereof. Described herein are ... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Lysine acetyltransferase 6a (kat6a) inhibitor, combinations and uses thereof. Described herein ar... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Crystalline methionine adenosyltransferase 2a (mat2a) inhibitor and uses thereof. Described herei... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Methionine adenosyltransferase 2a (mat2a) inhibitor combinations and uses thereof. Described here... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Nlrp3 inflammasome inhibitors and uses thereof. Described herein are NLRP3 inflammasome inhibitor... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Inhibitors of fgfr2 and fgfr3 and uses thereof. Described herein are FGFR2 and FGFR3 inhibitors a... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Cdk8/19 dual inhibitors and methods of use thereof. The disclosure provides for compounds and met... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Pro inhibitors for treating coronavirus infections. Provided herein are compounds, pharmaceutical... | 
				    				
				    			
				    				
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				    							G/S
				    						
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				    					Downloadable and recorded computer software; recorded or downloadable computer software platforms... | 
				    				
				    			
				    				
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				    							G/S
				    						
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				    					Downloadable computer software applications for estimating the relative binding free energy to pr... | 
				    				
				    			
				    				
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				    							Invention
				    						
				    						
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				    					Inhibitors of kif18a and uses thereof. Described herein are KIF18A inhibitors and pharmaceutical ... |