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2008
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Invention
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Modulators of urotensin receptor and methods of use thereof. Provided are compounds that are modu... |
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Invention
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Quinoline urotensin-ii receptor antagonists. Provided are compounds that are modulators of uroten... |
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Invention
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Thiophene-2-carboxamide derivatives as modulators of ccr9 receptor. Provided are compounds of For... |
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Invention
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Modulators of ccr9 receptor and methods of use thereof. Provided are compounds that are modulator... |
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Invention
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Formulations of n-(2-acetyl-4,6-dimethylphenyl)-3-{[(3,4 dimethyl-5-isoxazolyl)amino]sulfonyl}-2-... |
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Invention
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Formulations of n-(2-acetyl-4,6-dimethylphenyl)-3--2-thiophenecarboxamide.
Provided herein are i... |
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Invention
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Methods an compositions for treatment of an interstitial lung disease. Provided herein are method... |
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2007
|
Invention
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Modulators of c3a receptor and methods of use thereof.
Provided are compounds that are modulator... |
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Invention
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Modulators of c3a receptor and methods of use thereof. Provided are compounds that are modulators... |
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Invention
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Processes for the preparation of 4-chloro-3-methyl-5-(2-(2-(6-methylbenzo[d][1,3]dioxol-5-yl)acet... |
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Invention
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Processes for the preparation of n-(2-acetyl-4,6-dimethylphenyl)-3-{[(3,4 dimethyl-5-isoxazolyl)a... |
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Invention
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Polymorphs of n-(2-acetyl-4,6-dimethylphenyl)-3-{[(3,4 dimethyl-5-isoxazolyl)-amino]sulfonyl}-2-t... |
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Invention
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N- (4-chl0r0-3-methyl-5-is0xaz0lyl) -2- [2-methyl-4, 5- (methylenedioxy) phenylacetyl] -thiophene... |
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Invention
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Crystalline n-(4-chloro-3-methyl-5-isoxazolyl)-2-[2-methyl-4.5-(methylenedioxy)phenylacetyl]-thio... |
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Invention
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Pyridine, pyrimidine, quinoline, quinazoline, and naphthalene urotensin-ii receptor antagonists. ... |
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Invention
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Methods and compositions for treatment of sleep apnea.
Provided herein are methods of treatment ... |
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Invention
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Methods and compositions for treatment of sleep apnea comprising administration of an endothelin ... |
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Invention
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Formulations of sitaxsentan sodium.
Provided herein are stable lyophilized and oral formulations... |
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Invention
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Methods and compositions for treatment of diastolic heart failure.
Provided herein are methods o... |
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Invention
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Formulations of sitaxsentan sodium. Provided herein are stable lyophilized and oral formulations ... |
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Invention
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Methods and compositions for treatment of diastolic heart failure. Provided herein are methods of... |
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Invention
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Polymorphs of n-(4-chloro-3-methyl-5-isoxazolyl)2-⏧2-methyl-4,5-(methylenedioxy) phenylacetyl&rsq... |
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2005
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Invention
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Carboxylic acid derivatives that inhibit the binding of integrins to their receptors. 1 is involved. |
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2004
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Invention
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Phenylenediamine urotensin-ii receptor antagonists and ccr-9 antagonists. The present invention r... |
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Invention
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Pyridine, pyrimidine, quinoline, quinazoline, and naphthalene urotensin-ii receptor antagonists..... |
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2003
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Invention
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Combination products with carboxylic acid derivatives that inhibit the binding of integrins to th... |
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Invention
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Sulfonamides and derivatives thereof that modulate the activity of endothelin. Thienyl-, furyl- a... |
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2001
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Invention
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Sulfonamides for treatment of endothelin-mediated disorders. Thienylsulfonamides and their pharma... |
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Invention
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Biphenylsulfonamides and derivatives thereof that modulate the activity of endothelin. Biphenylsu... |
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Invention
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Propanoic acid derivatives that inhibit the binding of integrins to their receptors. A compound o... |
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Invention
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Method of treating glaucoma. Methods, compositions, and compounds for modulating the activity of ... |
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Invention
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Substituted phenyl compounds and derivatives thereof that modulate the activity of endothelin. Me... |
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Invention
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Formulation of sulfonamides for treatment of endothelin-mediated disorders. Formulations of pharm... |
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2000
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Invention
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Sulfonamides and derivatives thereof that modulate the activity of endothelin. Thienyl-, furyl-, ... |
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Invention
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Benzenesulfonamides and the use thereof to modulate the activity of endothelin. N-(5-isoxazolyl)b... |
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Invention
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Sulfonamides for treatment of endothelin-mediated disorders. Thienyl-, furyl- and pyrrolyl-sulfon... |
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1999
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Invention
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N-alkyl, n-alkenyl, n-alkynyl, n-aryl and n-fused bicyclo or tricyclo thienyl-, furyl-,and pyrrol... |
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1998
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Invention
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Phosphoramidates, phosphinic amides and related compounds and the use thereof to modulate the act... |
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1997
|
Invention
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N-aryl thienyl-, furyl-, and pyrrolyl-sulfonamides and derivatives thereof that modulate the acti... |
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Invention
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N-heteroaryl aryl-substituted thienyl-furyl-and pyrrolyl-sulfonamides and derviatives thereof tha... |
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1996
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Invention
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Process to inhibit binding of the integrin α4β1 , to vcam-1 fibronectin and cyclic peptides there... |
